5CR5 - X-RAY CRYSTAL STRUCTURE AT 1.61A RESOLUTION OF HUMAN MITOCHONDRIAL BRANCHED CHAIN AMINOTRANSFERASE (BCATM) COMPLEXED WITH A BIPHENYL PYRROLIDINE ETHER COMPOUND AND AN INTERNAL ALDIMINE LINKED PLP COFACTOR.

Hongfeng Deng; Jingye Zhou; Flora S. Sundersingh; Jennifer Summerfield; Don Somers; Jeffrey A. Messer; Alexander L. Satz; Nicolas Ancellin; Christopher C. Arico-Muendel; Katie L. (Sargent) Bedard; Arthur Beljean; Svetlana L. Belyanskaya; Ryan Bingham; Sarah E. Smith; Eric Boursier; Paul Carter; Paolo A. Centrella; Matthew A. Clark; Chun-wa Chung; Christopher P. Davie; Jennifer L. Delorey; Yun Ding; G. Joseph Franklin; LaShadric C. Grady; Kenny Herry; Clare Hobbs; Christopher S. Kollmann; Barry A. Morgan; Laura J. (Pothier) Kaushansky; Quan Zhou
PDBJ - 5CR5
https://pdbj.org/mine/summary/5cr5

Abstract

Branched-chain-amino-acid aminotransferase, mitochondrial, PYRIDOXAL-5'-PHOSPHATE, 3-({(3R)-1-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}oxy)-N-methyl-2'-[(methylsulfonyl)amino]biphenyl-4-carboxamide

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